Prostamax a bioengineered inoshanda peptide yakagadzirirwa kurapa dzakasiyana siyana dzeprostate zvirwere.
Yakagadziridzwa kuburikidza neyakakura mamorekuru-level research mu pathological nzira dzekusagadzikana uku, inobatanidza mitsetse yezvikamu kubva kune chaiyo kukura zvinhu, anti-inflammatory peptides, kana chiratidzo-modulating peptides.
Amino acid inotsiva, kutevedzana truncation, uye cyclization inoshandiswa kuwedzera kugadzikana kwayo, bioavailability, uye kunanga; kuderedzwa mukudzikira uye nekudaro hafu yeupenyu yakarebesa mibairo yakananga yeichi chiitiko.
Chiito chakananga pamatishu eprostate chinowanikwa.
Pakazara, Prostamax inomiririra multi-mechanism, synergistic bioactive mhinduro yekuvandudza murume prostate physiological hutano.
Kutevedzana
Lys-Glu-Asp-Pro
Nhamba yeCAS
/
Molecular Formula
C20H33N5O9
Molecular Weight
487.51
Tsvagiridzo yeProstamax Peptide
1.Maitiro Ekuita uye Kurapa Migumisiro
Kudzivirira nzira dzakakosha dzekuzvimba mukati me prostate pachayo ndeimwe yenzira dzayo dzekutanga dzekushanda – zvakakosha zvinoputika zvinhu zvinoratidzira zvakanyanya kudzvinyirirwa kutaura.
Kubudirira kuderedzwa kwemarudzi ose emamiriro ekuputira, kuzvimba kwakabatana uye kurwadziwa kunotevera, ensue.
Modulation of androgen receptor kuisa chiratidzo (kana pesvedzero yakananga pa 5α-reductase chiitiko) inogadzirisa DHT (Dihydrotestosterone) production (iyo yakanyanya simba fomu ye testosterone) uye zvinobudirira kudzora epithelial cell kuwanda.
Kuwedzera kuwanda kunokonzerwa neDHT isina kunyoreswa saka inodziviswa, zviratidzo zvepazasi weti (LUTS) kuva chikonzero chakananga chekuwedzera kweprostate.
Zvidzidzo zvakaratidzawo zvakakosha mukana weProstamax mukusimudzira apoptosis yemasero eprostate, angiogenesis inhibition, uye yakazara antioxidant / anti-inflammatory defense systems.
2.Kugadzirisa Hormonal Pathways
Sezvataurwa pamusoro apa, kutendeuka kwe testosterone kuDHT kwakakosha pakuita kwayo.
Aberrant kuwanda kunodzoserwa zvakanyanya nekuita uku.
3.Anti-inflammatory uye Antioxidant Migumisiro
The ambotaurwa kuzvimba uye oxidative kukuvara inoderedzwa.
4.Anti-Proliferative Basa
Kusungwa kwesero (G1 chikamu) inoratidzirwa maitiro ekurapa kweProstamax, uye semugumisiro wezvose zviri pamusoro, akadzorerwa physiological mamiriro eprostate inogona kuwanikwa.
Kudzvinyirira paurethra uye dundira, uye zviratidzo zvinosanganiswa zvechirwere chisingaperi, kurerukirwa.
COA
HPLC
MS





