Hexapeptide-2, atawa leuwih ilahar disebut GHRP-6, mangrupa α-melanocyte-stimulating hormone antagonis. Ngahambat tirosinase kagiatan, eta suppresses duanana produksi jeung déposisi saterusna pigmén; ngaronjatkeun nada kulit sakabéh mangrupa salah sahiji épék primér na.
The incorporation tina D-amino asam dina strukturna sacara signifikan ningkatkeun stabilitas métabolik, babarengan jeung strengthened reséptor mengikat stabilitas jeung pangirut. Sacara stuktur sami sareng α-MSH sorangan, Hexapeptide-2 ngahalangan kamampuan hormon ieu pikeun ngabeungkeut na reséptor – melanosit kagiatan jadi target langsung dihambat.
Salaku hiji sarua GHRP-6, pulsatil hipofisis sékrési tina hormon pertumbuhan dirangsang; sintésis protéin, ngembangkeun tulang (sareng sadaya prosés perbaikan anu aya hubunganana), nyageurkeun tatu, sareng ningkatkeun fungsi imun sadayana dipangaruhan sacara positif.
Runtuyan
Na-Trp-Ala-Trp-Phe-Lys atanapi H-His-D-Trp-Ala-Trp-D-Phe-Lys-NH2
Nomer CAS
87616-84-0
Formula Molekul
C46H56N12O6
Beurat Molekul
873.014
Hexapeptide-2 Panalungtikan patali
1.Poténsi Aplikasi Terapi
poténsi cosmetological ngajangjikeun aya salaku agén whitening atawa terapi pikeun sagala rupa wangun hiperpigmentasi gangguan. Sipat antagonis ogé nyarankeun panggunaan poténsi anu langkung lega: stimulasi napsu, cachexia perbaikan, sareng modulasi peradangan.
2.Antagonis jalur sinyal α-MSH
Beungkeutan reséptor kompetitif mangrupikeun mékanisme konci; ngurangan mélanin sintésis mangrupa hasil langsung.
Lightening kulit éféktif mangrupa hasil ahir prosés ieu. Puseur napsu di hipotalamus bisa dipangaruhan, kalayan perbaikan kualitas kahirupan pikeun penderita cachexia atanapi leungitna napsu anu aya hubunganana sareng umur janten kauntungan sekundér anu berharga.
3.Promoting Pulsatile Growth Hormone Secretion
Synergistic enhancement of endogenous ghrelin and suppression of somatostatin are what drive the desired pulsatile release.
This physiological pattern of release is considered a more effective therapeutic approach to avoid desensitization.
4.Stimulating Tissue and Bone Repair
Increased levels of growth hormone and IGF-1 promote mitotic and anabolic kagiatan, thereby stimulating tissue proliferation, diferensiasi, and repair.
This accelerates the repair of soft tissue and bone, promotes fibroblast proliferation and kolagén sintésis, and enhances wound healing.
Sajaba, it stimulates osteoblast activity and bone matrix formation, which helps increase bone density, accelerate fracture healing, and combat age-related bone loss.
COA
HPLC
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