Hexapeptide-2, ko fiye da ake kira da GHRP-6, wani ne α-melanocyte-stimulating hormone antagonist. Hana tyrosinase aiki, yana hana duka samarwa da kuma shigar da pigment na gaba; inganta sautin fata gaba ɗaya yana ɗaya daga cikin tasirin sa na farko.
Haɗin kai na D-amino acid a cikin tsarinsa yana haɓaka kwanciyar hankali na rayuwa, tare da ƙarfafa mai karɓa mai ɗaure kwanciyar hankali da kusanci. Tsari yayi kama da α-MSH kanta, Hexapeptide-2 yana toshe ikon wannan hormone don ɗaure shi masu karɓa – melanocyte ayyuka kasancewar an hana niyya kai tsaye.
A matsayin daidai da GHRP-6, bugun jini pituitary asiri na girma hormone yana kara kuzari; gina jiki kira, ci gaban kashi (da duk hanyoyin gyarawa masu alaƙa), warkar da rauni, da haɓaka aikin rigakafi duk suna da tasiri mai kyau.
Jeri
His-Trp-Ala-Trp-Phe-Lys ko H-His-D-Trp-Ala-Trp-D-Phe-Lys-NH2
Lambar CAS
87616-84-0
Tsarin kwayoyin halitta
Saukewa: C46H56N12O6
Nauyin Kwayoyin Halitta
873.014
Hexapeptide-2 Bincike mai alaƙa
1.Aikace-aikace masu yuwuwar warkewa
Alkawari cosmetological m wanzu a matsayin whitening wakili ko warkewa ga daban-daban siffofin hyperpigmentation cuta. Abubuwan da ke gaba da juna kuma suna ba da shawarar fa'idar amfani: sha'awar ci, cachexia inganta, da daidaita yanayin kumburi.
2.adawa hanyar siginar α-MSH
Haɗin mai karɓar gasa shine maɓalli mai mahimmanci; ragewa melanin kira shine sakamako kai tsaye.
Ingantacciyar walƙiyar fata shine ƙarshen sakamakon wannan tsari. Cibiyoyin ci a cikin hypothalamus ana iya yin tasiri, tare da ingancin inganta rayuwa ga marasa lafiya tare da cachexia ko asarar ci da ke da alaƙa da shekaru kasancewa wata fa'ida ta biyu mai mahimmanci.
3.Haɓaka Sirin Hormone na Ci gaban Pulsatile
Haɓaka haɗin gwiwa na endogenous ghrelin da kuma danne somatostatin su ne abin da ke fitar da bugun bugun jini da ake so.
Ana ɗaukar wannan tsarin sakin jiki a matsayin mafi inganci hanyar warkewa don guje wa rashin jin daɗi.
4.Gyaran Nama da Ƙashi Mai Ƙarfafawa
Ƙara yawan matakan hormone girma da Farashin IGF-1 inganta mitotic da anabolic aiki, ta haka yana kara kuzari yaduwa, bambanta, da gyarawa.
Wannan yana hanzarta gyaran nama mai laushi da kashi, inganta fibroblast yaduwa da collagen kira, kuma yana inganta warkar da raunuka.
Bugu da kari, yana kara kuzari osteoblast aiki da samuwar matrix kashi, wanda ke taimakawa wajen kara yawan kashi, hanzarta karaya waraka, da yaki da asarar kashi mai alaka da shekaru.
COA
HPLC
MS





