Adamax na roba ne heptapeptide samu daga ban ji ba; takamaiman jerin amino acid shine Ac-MEHFPG-AG-NH₂.
Semax kanta, gutsure na adrenocorticotropic hormone (ACTH), yana da tasiri mai ƙarfi na neurotrophic da haɓaka fahimi.
Ƙayyadaddun tsari a cikin jima'i yana haifar da iyakacin iyaka ga rabin rayuwar sa da ingancin ketare shingen kwakwalwar jini..
Don rage waɗannan gazawar masana kimiyya sun gabatar da babbar ƙungiyar adamantylacetate ta hanyar covalent bonding a cikin tashar carboxyl.
Wannan gyara ya inganta sosai pharmacokinetic Properties na kwayoyin peptide.
Gabatarwar wannan rukunin yana ba da cikakkiyar juriya ga na gaba lalacewar enzymatic; lokacin riƙewa na nau'in aiki na adamax a cikin jiki yana da tsawo sosai.
Mai ban sha'awa, wanda aka ambata a baya ‘masu hankali’ ƙira yana haɓaka haɓakar haɓakawa wanda peptide ke ƙetare ya ce shinge, kuma ana samun ƙayyadaddun ƙayyadaddun ƙayyadaddun ƙima da zaɓi.
Rashin daidaituwa ba ayyukan ilimin halitta, duk sanannun tasirin semax ana kiyaye su ko haɓakawa.
Jeri
Ac-MEHFPGP-Adam-NH2
Lambar CAS
/
Tsarin kwayoyin halitta
Saukewa: C50H68N10O12S
Nauyin Kwayoyin Halitta
1033.212
Binciken Adamax:
1.Ingantaccen Maganin warkewa da Yiwuwar Clinical
Gwaje-gwaje na asibiti sun nuna Adamax don haɓaka Semax a cikin haɓaka haɓaka da kariyar Neurotrophic factor na kwakwalwa da aka samu (BDNF) kuma zuwa wani batu jijiya girma factor (NGF).
Maye gurbin Semax azaman wakili na warkewa, musamman ga cututtukan hauka ko haɓaka fahimtar zamantakewa, yuwuwar gaske ce.
2.Haɓaka Hankali (Hankali kasancewar sashe ne)
Ƙarfafa kai tsaye na haɓakar BDNF shine babban aikin Adamax.
Ayyukan ƙwayoyin jijiyoyi, sabon ƙarni na neuron / bambance-bambancen da duk abubuwan haɓaka synaptic da ke da alaƙa shine abin da bincike ke mayar da hankali kan yanzu.
Ayyukan hippocampal da prefrontal cortex suma sun karu.
Ƙungiyoyin gwaji na dogon lokaci suna da kuma za su ci gaba da nunawa, adadi, mafi girman ƙwaƙwalwar ajiya da ƙwarewar koyo.
3.Tasirin Neuroprotective
Haɓaka fahimi na Adamax da ayyukan haɓaka hankali sun samo asali ba kawai daga haɓakar haɓakar ƙwayoyin jijiyoyi kai tsaye ba., amma kuma daga abubuwan da ake iya gani na neuroprotective.
An nuna ingantacciyar raguwar wuraren ɓarna a cikin marasa lafiya na bugun jini; ƙarfafawa da dawo da ƙwayoyin necrotic daban-daban shine wani muhimmin al'amari na wannan neuroprotection.
Ragewa excitotoxicity da kuma samar da tasirin antioxidant na kusa-kusa yana da ƙari, ayyuka masu kyau da aka rubuta.
Matsayi kanta a cikin wannan daula, Adamax yana ɗaukar alƙawarin da yawa azaman wakili na warkewa na gaskiya don cututtukan neurodegenerative – Alzheimer shine babban misali, Parkinson yana biye a baya.
4.Damuwa da Rage damuwa
Adamax yana haɓaka ikon ɗan adam don dacewa da canje-canjen muhalli; kwakwalwa kanta dole ne cikin sauri daidaita zuwa, da tsayayya, iri-iri na matsalolin physiological da ke haifar da waɗannan sauye-sauyen yanayi mai sauri.
Kula da wani nau'i na homeostasis shine makasudin ƙarshe.
Modulation na hypothalamic-pituitary-adrenal (HPA) axis shine tsakiyar wannan tsari, karuwa ko rage sakin da ya dace na neurotransmitters, duk kankantar martanin ‘danniya’ ana danne.
Anxiolytic Tasiri shine fa'ida ta farko – drowsiness da rashin fahimta (illolin da ke kusa da duniya na anxiolytics na gargajiya) ana kaucewa gaba daya.
Haɓaka aikin fahimi yayin kowane nau'i na taimako na damuwa shine abin da ke sa Adamax ya zama abin sha'awa ga masu bincike da marasa lafiya iri ɗaya..
COA
HPLC
MS





