Prostamax bụ a bioengineered peptide na-arụ ọrụ emebere maka ọgwụgwọ ọrịa prostate dị iche iche.
Emepụtara site na nyocha ọkwa ọkwa dị ukwuu n'ime pathological usoro nke nsogbu ndị a, ọ na-agụnye usoro akụkụ ụfọdụ sitere na kpọmkwem ihe na-eto eto, mgbochi mkpali peptides, ma ọ bụ peptides na-agbanwe mgbaàmà.
Amino acid nnọchi, usoro nkwụsịtụ, na cyclization na-eji mee ka ọ kwụsie ike, bioavailability, na ezubere iche; Mbelata nbibi na ya mere ogologo ndụ ọkara ndụ ogologo bụ nsonaazụ nke usoro a.
A na-eme ihe kpọmkwem na anụ ahụ prostate.
N'ozuzu, Prostamax na-anọchite anya ọtụtụ usoro, Ihe ngwọta bioactive synergistic iji meziwanye ahụ ike physiological nwoke prostate.
Usoro
Lys-Glu-Asp-Pro
Nọmba CAS
/
Usoro ihe omimi
C20H33N5O9
Ibu molekụla
487.51
Nnyocha nke Prostamax Peptide
1.Usoro nke Omume na Mmetụta Ọgwụgwọ
Mgbochi ụzọ mgbama mkpasu iwe n'ime prostate n'onwe ya bụ otu n'ime ụdị ọrụ ya bụ isi – ihe mkpali dị egwu na-egosipụta nkwubi okwu ebelatara nke ukwuu.
Mbelata nke ọma nke ụdị ọ bụla nke ọnọdụ mkpali, ọzịza jikọtara na mgbu na-esote, sonye.
Mgbanwe nke androgen receptor na-egosi (ma ọ bụ kpọmkwem mmetụta na 5α-reductase ọrụ) na-achịkwa DHT (Dihydrotestosterone) mmepụta (ụdị testosterone dị ike karị) ma na-achịkwa mgbasa nke cell epithelial nke ọma.
A na-egbochi mmụba dị ukwuu nke DHT na-akwadoghị, obere mgbaàmà urinary tract (LUTS) ịbụ ihe sitere na prostate ịgbatị.
Nnyocha egosiwokwa nnukwu ikike maka Prostamax n'ịkwalite apoptosis nke sel prostate, mgbochi nke angiogenesis, yana usoro nchekwa ihe mgbochi / mgbochi mkpali zuru oke.
2.Na-achịkwa usoro Hormonal
Dị ka e kwuru n'elu, ntughari nke testosterone na DHT bụ ihe dị mkpa na omume ya.
Usoro a na-agbanwe nke ukwuu n'ịba ụba nke aberrant.
3.Mmetụta mgbochi mkpali na Antioxidant
Nke e kwuru n'elu mkpali na mmebi oxidative na-ebelata.
4.Ọrụ mgbochi-Proliferative
Ejide okirikiri cell (Akụkụ G1) bụ egosipụtara mmetụta nke ọgwụgwọ Prostamax, na n'ihi ihe niile dị n'elu, enwere ike nwetaghachi ọnọdụ physiological nke prostate.
Nrụgide na urethra na eriri afo, na ihe mgbaàmà metụtara ọrịa na-adịghị ala ala, na-enwe ahụ iru ala.
COA
HPLC
MS





