Testagen ke peptide ea maiketsetso e sebetsang ka bongata e nkiloeng lipatlisisong tse fapaneng tsa kalafo ea peptide le taolo ea endocrine..
Liphetoho tsa biomimetic tse thehiloeng ho li-peptide tsa tlhaho, hammoho le lipapiso tsa limolek'hule tse thusoang ke k'homphieutha, li sebelisitsoe ho matlafatsa botsitso le bioavailability ea eona; Ka mor'a moo, immunogenicity ea fokotseha.
Liphuputso tsa pele li bontša hore Testagen e susumetsa hypothalamic-pituitary-gonadal axis, laolang testosterone secretion ka ho khetheha.
Ts'ebetso ea AMPK le tse fapa-fapaneng sirtuin pontsho litselana latela, e khothalletsa ho kenngoa ha mafura a acid le glucose – ho bokellana ha mafura a visceral le profiles ea lipid ka kakaretso e le lintlafatso tsa bohlokoa tse bonoang.
Teko, Ka kakaretso, ke sethethefatsi sa 'nete sa maiketsetso sa peptide se nang le sepheo se ngata; mafu a amanang le metabolic le lilemo a ka fihlella boemo ba ona ba ts'ebetso.
Tatelano
H-Lys-Glu-Asp-Gly-OH
Nomoro ea CAS
1026993-38-3
Foromo ea limolek'hule
C17H29N5O9
Boima ba Molek'hule
447.445
Lipatlisiso tsa Testagen Peptide
1.Liphello tsa Metabolic le Neurological
Bopaki ba liteko tsa tlase K'holeseterole ea LDL le triglycerides e teng; mofuta 2 kalafo ea lefu la tsoekere ke e 'ngoe ea ts'ebeliso e ka bang teng.
Liphuputso tsa morao tjena li senotse matla a bohlokoa a antioxidant (har'a liphello tse ling), matlafatsa superoxide dismutase le glutathione peroxidase mosebetsi, phokotso ea mefuta eohle ea oxidative cell necrosis joalo ka sepheo sa moleng ona oa lipatlisiso.
Haholo-holo lipatlisiso li bontša hore li ntlafetse mitochondrial tshebetso.
Ho tšela mokoallo oa mali bokong, Testage e susumetsa boko bo nkiloeng ke neurotrophic factor (BDNF) sephiri; ts'ebetso ea kelello le ho phela ha neuronal ka bobeli li ameha hantle.
2.Matlafatso ea Endocrine
Ho feto-fetoha ha lets'oao le boletsoeng ka holimo ke sepheo sa mantlha.
Ka ho toba, taolo e nepahetseng ea tsamaiso ea endocrine boemong ba pontšo ke eona e etsang hore Testagen e hlokomelehe ka ho khetheha.
Ho etsisa tokollo ea Hormone e lokollang gonadotropin(GnRH) ka har'a hypothalamus, optimization ea secretion ea pituitary (ea bonyane Hormone ea luteinizing /LH) finyelloa.
Pontšo ea liprotheine tse matla (e amanang le steroidogenesis liseleng tsa testicular) e ka boela ea fetoloa, phepelo ea matla a mitochondrial joalo ka ntlha ea bobeli empa e le ea bohlokoa.
Ho fokotsa 'mele’ ea globulin e tlamang lihomone tsa thobalano (SHBG) bakeng sa testosterone ke tsela e 'ngoe eo Testagen e e nkang ho finyella phetoho ea endocrine.
Tsena tsohle li kopane, bolokehileng (ho tsebo ya jwale) kalafo e thehiloeng ho endocrine kapa bonyane likarolo tsa eona, li 'me e tla lula e le karolo ea tšepiso ea kalafo ea Testagen.
3.Taolo ea Matla
Testagen e kenya tšebetsong AMP-activated protein kinase pathway kapa AMPK, mofuta oa cellular 'energy switch'.
Ho etsisa pontšo ena, e khothalletsa oxidation ea mafura a mafura ka har'a sebete le mesifa ea mesifa, e thibela mefuta e fapaneng ea lipid synthesis.
Ho hatella triglycerides le low-density lipoprotein ke phello e tobileng ea ketso ena.
Ho matlafatsa kutloisiso ea insulin ke phello e 'ngoe ea bohlokoa; Tšebeliso ea matla a lisele le litho tsa 'mele e ea ntlafatsoa, ho hanyetsa insulin ho fokotsehile haholo – ho bokella mafura a masoeu a visceral e le e 'ngoe ea lintlha tse ka lekanyetsoang tsa ts'ebetso ena.
Taolo e pharalletseng ea matla ke eona e sebetsanang le botenya le bofokoli bohle bo amanang le tsoekere ea mali bo bakoang ke lijo tse mafura a mangata.; boleng ba kalafo bo ka bang teng bakeng sa mofuta 2 lefu la tsoekere le ngotsoe hantle.
4.Liphello tsa Antioxidant
Liphuputso li bonts'a Testagen e ntlafatsa ts'ebetso ea bonyane li-enzyme tse amanang le antioxidant (catalase, glutathione peroxidase joalo ka moemeli), ho sutumelletsa moeli o kaholimo oa sistimi ea ts'ireletso ea 'mele ea antioxidant.
Matla a bohlokoa a tlhaho a ho itšireletsa mafung aa matlafatsoa, tshenyo e fokolang ea oxidative liseleng ka bobeli le (ho isa tekanyong e kgolo) DNA e etsahala.
Lipatlisiso tse khahlanong le botsofali li bontšitse ka ho khetheha ho fokotseha ha mitochondrial, telomere attrition le likarolo tsohle tse nyane tsa boleng ba ho phela ha lisele – motheo o tiileng oa theory bakeng sa kopo efe kapa efe e khahlanong le botsofali.
Liphello tsa Ntlafatso ea Neuroprotective le Cognitive: Testagen ke peptide e entsoeng ka hloko e etselitsoeng ho tšela mokoallo oa boko ba mali.
Modulating Moamoheli oa NMDA ts'ebetso ke ts'ebetso ea eona ea mantlha e reriloeng ke neuroprotective.
Boko bo entsoeng ke neurotrophic factor (BDNF) synthesis le mekhoa e amanang le eona – pholoho, karohano le kholo e kholo ea methapo ea kutlo – e boetse e susumetsoa.
Neurogenesis ka har'a hippocampus, kholiso ea mohopolo le mathata ohle a amanang le kelello a ntlafatsoa.
Ho fokotsa β-amyloid mofuta oa chefo le tahlehelo ea dopaminergic neurons (le tsohle tse latelang ‘ho shoa morao’ ya boko) e etsa ntlha e batloang ea ho qetela ea lipatlisiso tsa neurodegenerative.
COA
HPLC
MOF





