Myristoyl Pentapeptide-4 ke peptide ea biofunctional e thusang ho boloka letlalo le tletse, ho tiea, le ponahalo ya botjha.
E entsoe ho ipapisitsoe le ho etsisa le kutloisiso e rarahaneng ea insulin-like growth factor-1 (IGF-1) le karolo ea eona ea ho laola ho ata ha lisele, karohano, apoptosis le synthesis ea matrix a extracellular lintho tse kang collagen le elastin.
IGF-1 ha e loketse tšebeliso ea litlolo ka lebaka la boima ba eona bo boholo ba molek'hule bo sitisang ho kenella ka har'a letlalo., botsitso bo futsanehileng le theko e phahameng. Ka ho hlahloba libaka tsa bohlokoa tsa li-receptor tsa IGF-1, tatellano ea mantlha ea Lys-Thr-Thr-Lys-Ser e ile ea khetholloa.
E boetse e bonts'a mamello e ntle letlalong le nang le kutloelo-bohloko 'me ka hona e fetohile karolo ea bohlokoa e sebetsang ho li-topical anti-ageing dermatological formulations..
Tatelano
Lys-Thr-Thr-Lys-Ser (KTTKS)
Nomoro ea CAS
1392416-25-9
Foromo ea limolek'hule
C37H71N7O10
Boima ba Molek'hule
774.00
Lipatlisiso tse amanang le Myristoyl Pentapeptide-4
1.Mokhoa oa Motheo le Liphello tsa mantlha
N-terminal myristoylation e ntlafalitse haholo lefu la tsoekere le ho phunyeletsa letlalo, ho nolofalletsa peptide ho tlama ka kotloloho ho li-receptor tsa IGF-1 le ho kenya tšebetsong lipontšo tse tlase.
Sena, ka mor'a moo, e tsosa ho fokotseha ho amanang le lilemo tsa anabolic cutaneous process; e phahamisa sekhahla sa tlhahiso ea mefuta e fapaneng ea liprotheine tsa matrix tsa extracellular tse kang Kenya mofuta oa collagen, Mofuta oa III oa collagen le elastin – ka mafolo-folo ho kgutlisa dermal cell degradation e bakoang ke botsofali.
Sena se eketsa haholo bongata le botenya ba lisele tsa dermal, e bontshang bokgoni bo matla ba ho fokotsa kapa ho hlakola makukuno a sa fetoheng.
2.E thusa ho Kopana ha Mofuta oa I le oa III oa Collagen
Collagen mofuta oa I le III ke liprotheine tse ka sehloohong tse khethollang letlalo le tiileng le ho tiea.
Bokhoni ba bona ba tlhaho ba tlhaho bo fokotseha haholo ka lilemo.
Myristoyl Pentapeptide-4 e sebetsa ka ho etsisa pontšo ea IGF-1, e tlamang ho insulin-like growth factor-1 receptor le ho kenya likarabo tsa anabolic ho fibroblasts.
Sena se eketsa tlhahiso ea collagen ea Mofuta oa I le oa III, e kokobetsang letlalo la letlalo ha e ntse e fokotsa mela e metle le masoebe a amanang le botsofali. 1
3.E matlafatsa Elastin Synthesis le Mokhatlo
Myristoyl Pentapeptide-4 e laola elastin polelo ea lefutso le tlhahiso ea protheine nakong ea ts'ebetso ea fibroblast.
E susumetsa liprotheine tse sa tsoa hlahisoa hore li hlophisehe ho ba marang-rang a laetsoeng a fiber, e matlafatsang letlalo le tshehetsang.
Sena se eketsa elasticity ea letlalo, ka potlako boreleli makukuno a bakoang ke tahlehelo ya tshehetso e ka hare, ha e ntse e sebetsana le ho fokotseha.
Boreleli ba letlalo hang-hang bo fetoha boreleli, ho ntlafatsa boemo ba letlalo ka kakaretso.
COA
HPLC
MOF





